结合停留时间和传统结合亲和力提供了一个更全面的框架,用于理解药物-靶点相互作用并指导合理的药物设计。优化停留时间可以增强药效学效能,提高靶点选择性,并提升安全性。因此,停留时间正成为现代药物发现中的关键动力学参数。
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Lu Liu
Zerong Xu
Dong Guo
Expert Opinion on Drug Discovery
Xuzhou Medical College
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Liu 等人(周三)研究了此问题。
www.synapsesocial.com/papers/6973106cc8125b09b0d20292 — DOI: https://doi.org/10.1080/17460441.2026.2619070
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