PulseExploreJournal ClubDebatesTrendingResearchersJournals
Instagram
HomeExploreJournal ClubTrending
Synapse
⌘+K
Synapse
March 29, 2026Chemistry & Biodiversity0 citationsOpen Access

Inhibitors of Sodium‐Dependent Serotonin Transporter Protein (SERT) as Potential New Nematicides

View Full Paper
GHGeraldo Jamisse HodelaVSVitor Pereira de SousaMMMariana Castro de Melo

Key Points

  • To evaluate SERT inhibitors as potential new nematicides against Meloidogyne nematodes.
  • Conducted in silico analysis to identify protein targets of chaetoglobosins A and B.
  • Evaluated SERT inhibitors' effectiveness in vitro against Meloidogyne juveniles.
  • Measured mortality rates using paroxetine and commercial nematicide fluensulfone.
  • Paroxetine achieved 50% mortality (LC50) at 351.3 µg/mL in Meloidogyne incognita.
  • Fluensulfone showed a lower LC50 of 39.3 µg/mL under the same conditions.
  • Paroxetine reduced the pathogenicity of Meloidogyne incognita juveniles during plant trials.

Abstract

Nematodes of the genus Meloidogyne cause major losses in agricultural production worldwide. To identify potentially useful chemical structures for developing new nematicides, this study initially aimed to determine in silico - using computationally efficient techniques - the protein target of chaetoglobosins A and B in these nematodes. This process led to the selection of the sodium-dependent serotonin transporter protein (SERT). The activities of SERT inhibitors were subsequently evaluated in vitro. The best result was obtained with paroxetine, which caused 50% mortality (LC50) in second-stage juveniles (J2) of Meloidogyne incognita at a concentration of 351.3 µg/mL. Under the same conditions, the commercial nematicide fluensulfone showed an LC50 of 39.3 µg/mL. In plant trials, paroxetine reduced the pathogenicity of M. incognita J2. Therefore, further investigation of SERT inhibitors holds promise for the development of new nematicides.

Ask AI
Helpful
Bookmark
Share
View Full Paper

Cite This Study

Hodela et al. (2026) studied this question.

synapsesocial.com/papers/69c8c2d1de0f0f753b39d497https://doi.org/10.1002/cbdv.202503443
Ask AI
Helpful
Bookmark
Share
View Full Paper