Functionalisation of homopropargyl boronic esters via hydrozirconation followed by Pd-catalysed cross coupling reaction

Puntos clave

• The aim is to explore the functionalisation of homopropargyl boronic esters using hydrozirconation and cross coupling.
• Utilization of hydrozirconation for reactive functionalisation.
• Application of Pd-catalysed cross coupling reactions.
• Synthesis of homopropargyl boronic esters via Matteson homologation.
• Successful selective functionalisation of homopropargyl boronic esters.
• Retention of boronic ester functionality during the reaction.

Resumen